James E Audia: search on Z-Library

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1

US immigration order strikes against biotech

Levin, Jeremy M, Holtzman, Steven H, Maraganore, John, Hastings, Paul J, Cohen, Ron, Dahiyat, Bassil, Adams, Julian, Adams, Chris, Ahrens, Brett, Albers, Jeff, Aspinall, Mara G, Audia, James E, Babler

Journal:

Nature Biotechnology

Year:

2017

Language:

english

File:

PDF, 133 KB

english, 2017

2

Biotech leaders call for free press

Cohen, Ron, Holtzman, Steven, Levin, Jeremy M, Maraganore, John M, Aberman, Michael, Adams, Chris, Adams, Julian, Albers, Jeffrey, Anderson, Bonnie, Aspinall, Mara G, Audia, James E, Babler, Martin, B

Journal:

Nature Biotechnology

Year:

2018

Language:

english

File:

PDF, 130 KB

english, 2018

3

Diving into the water: Inducible binding conformations for BRD4, TAF1(2), BRD9, and CECR2 bromodomains

Crawford, Terry D., Tsui, Vickie, Flynn, E. Megan, Wang, Shumei, Taylor, Alexander M., Côté, Alexandre, Audia, James E., Beresini, Maureen H., Burdick, Daniel J., Cummings, Richard T., Dakin, Les A.,

Journal:

Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 1.94 MB

english, 2016

4

Synthesis of the individual enantiomers of the benzoquinolinone human type 1 steroid 5-α-reductase inhibitors LY191704 and LY266111

James E. Audia, David E. Lawhorn, Jack B. Deeter

Journal:

Tetrahedron Letters

Year:

1993

Language:

english

File:

PDF, 297 KB

english, 1993

5

Characterization of type I 5α-reductase activity in DU145 human prostatic adenocarcinoma cells

Kaefer, Martin, Audia, James E., Bruchovsky, Nicholas, Goode, Robin L., Hsiao, Kenneth C., Leibovitch, Ilan Y., Krushinski, Joseph H., Lee, Chung, Steidle, Christopher P., Sutkowski, Debra M., Neubaue

Journal:

The Journal of Steroid Biochemistry and Molecular Biology

Year:

1996

Language:

english

File:

PDF, 926 KB

english, 1996

6

Corrigendum to “Development of methyl isoxazoleazepines as inhibitors of BET” [Bioorg. Med. Chem. Lett. 25/9 (2015) 1842–1848]

Hewitt, Michael C., Leblanc, Yves, Gehling, Victor S., Vaswani, Rishi G., Côté, Alexandre, Nasveschuk, Christopher G., Taylor, Alexander M., Harmange, Jean-Christophe, Audia, James E., Pardo, Eneida,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 175 KB

english, 2015

7

Central and peripheral pharmacodynamic effects of BACE1 inhibition following oral administration of LY2811376 to PDAPP mice and beagle dog

May, Patrick C., Boggs, Leonard N., Yang, Zhixiang, Lindstrom, Terry, Calligaro, David, Citron, Martin, Sheehan, Scott, Audia, James E.

Journal:

Alzheimer's & Dementia

Year:

2010

Language:

english

File:

PDF, 62 KB

english, 2010

8

Early Drug Discovery Efforts Towards the Identification of EP300/CBP Histone Acetyltransferase (HAT) Inhibitors

Wilson, Jonathan Edward, Huhn, Annissa, Gardberg, Anna S., Poy, Florence, Brucelle, Francois, Vivat, Valerie, Patel, Gaurav, Patel, Chirag, Cummings, Richard, Sims, Robert, Levell, Julian, Audia, Jame

Journal:

Year:

2020

Language:

english

File:

PDF, 1.97 MB

english, 2020

9

Amyloid β-Mediated Oxidative and Metabolic Stress in Rat Cortical Neurons: No Direct Evidence for a Role for H2O2 Generation

Zhiyuan Zhang, Russell E. Rydel, Gary J. Drzewiecki, Kimberly Fuson, Sarah Wright, Mark Wogulis, James E. Audia, Patrick C. May, Paul A. Hyslop

Journal:

Journal of Neurochemistry

Year:

1996

Language:

english

File:

PDF, 1.31 MB

english, 1996

10

Development of methyl isoxazoleazepines as inhibitors of BET

Hewitt, Michael C., Leblanc, Yves, Gehling, Victor S., Vaswani, Rishi G., Côté, Alexandre, Nasveschuk, Christopher G., Taylor, Alexander M., Harmange, Jean-Christophe, Audia, James E., Pardo, Eneida,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 726 KB

english, 2015

11

Kidney disease in patients with obesity: It is not always obesity-related glomerulopathy alone

Salvatore, Steven P., Chevalier, James M., Kuo, Sheng F., Audia, Pat F., Seshan, Surya V.

Journal:

Obesity Research & Clinical Practice

Year:

2017

Language:

english

File:

PDF, 2.79 MB

english, 2017

12

GNE-371, a Potent and Selective Chemical Probe for the Second Bromodomains of Human Transcription-Initiation-Factor TFIID Subunit 1 and Transcription-Initiation-Factor TFIID Subunit 1-like

Wang, Shumei, Tsui, Vickie, Crawford, Terry D., Audia, James E., Burdick, Daniel J., Beresini, Maureen H., Côté, Alexandre, Cummings, Richard, Duplessis, Martin, Flynn, E. Megan, Hewitt, Michael C., H

Journal:

Journal of Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 4.65 MB

english, 2018

13

Jump rope rotation in trans-cycloalkenes

James A. Marshall, Vicki H. Audia, Todd M. Jenson, Wayne C. Guida

Journal:

Year:

1986

Language:

english

File:

PDF, 907 KB

english, 1986

14

Total synthesis of the Fusarium toxin equisetin: proof of the stereochemical relationship of the tetramate and terpenoid sectors

Turos, Edward, Audia, James E., Danishefsky, Samuel J.

Journal:

Journal of the American Chemical Society

Year:

1989

Language:

english

File:

PDF, 798 KB

english, 1989

15

Identification of EZH2 and EZH1 Small Molecule Inhibitors with Selective Impact on Diffuse Large B Cell Lymphoma Cell Growth

Garapaty-Rao, Shivani, Nasveschuk, Christopher, Gagnon, Alexandre, Chan, Eric Y., Sandy, Peter, Busby, Jennifer, Balasubramanian, Srividya, Campbell, Robert, Zhao, Feng, Bergeron, Louise, Audia, James

Journal:

Chemistry & Biology

Year:

2013

Language:

english

File:

PDF, 2.01 MB

english, 2013

16

Additions and Corrections - Acyclic Stereocontrol in Catalyzed Intramolecular Diels-Alder Cyclizations of 4-Methyl-2,8,10-undecatrienals.

Marshall, James, Audia, James, Grote, Jonathon

Journal:

Journal of Organic Chemistry

Year:

1986

Language:

english

File:

PDF, 134 KB

english, 1986

17

Resolution of δ-Lactams Provides Access to Nonracemic Benzoquinolinones: The Synthesis of LY300502 and LY300503

Astleford, Bret A., Audia, James E., Deeter, Jack, Heath, Perry C., Janisse, Samantha K., Kress, Thomas J., Wepsiec, James P., Weigel, Leland O.

Journal:

Journal of Organic Chemistry

Year:

1996

Language:

english

File:

PDF, 294 KB

english, 1996

18

Intramolecular Diels-Alder cyclization of conjugated aldehydes. Synthesis of a chlorothricolide intermediate

Marshall, James A., Audia, James E., Grote, Jonathan

Journal:

Journal of Organic Chemistry

Year:

1984

Language:

english

File:

PDF, 408 KB

english, 1984

19

Conjugate addition of organocuprates to trans-4a,5,6,7,8,8a-hexahydronaphthalene-1-carboxaldehydes. Synthesis of a chlorothricin degradation product

Marshall, James A., Audia, James E., Shearer, Barry G.

Journal:

Journal of Organic Chemistry

Year:

1986

Language:

english

File:

PDF, 911 KB

english, 1986

20

UNRESOLVED ISSUES IN DIALYSIS: Extracorporeal Strategies for the Removal of Middle Molecules

James F. Winchester, Patrick F. Audia

Journal:

Seminars in Dialysis

Year:

2006

Language:

english

File:

PDF, 100 KB

english, 2006

21

Synthesis of some 3-(1-azabicyclo[2.2.2]octyl) 3-amino-2-hydroxy-2-phenylpropionates: profile of antimuscarinic efficacy and selectivity

Audia, Vicki H., McPherson, Daniel W., Weitzberg, Moshe, Rzeszotarski, W. Janusz, Sturm, Bonnie, Kachur, James F., Abreu, Mary, Kaiser, Carl

Journal:

Journal of Medicinal Chemistry

Year:

1990

Language:

english

File:

PDF, 527 KB

english, 1990

22

Metformin-induced lactic acidosis and acute pancreatitis precipitated by diuretic, celecoxib, and candesartan-associated acute kidney dysfunction

Audia, Pat, Feinfeld, Donald A., Dubrow, Alan, Winchester, James F.

Journal:

Clinical Toxicology (Informa Healthcare)

Year:

2008

Language:

english

File:

PDF, 52 KB

english, 2008

23

Corrigendum: The promise and peril of chemical probes

Arrowsmith, Cheryl H, Audia, James E, Austin, Christopher, Baell, Jonathan, Bennett, Jonathan, Blagg, Julian, Bountra, Chas, Brennan, Paul E, Brown, Peter J, Bunnage, Mark E, Buser-Doepner, Carolyn, C

Journal:

Nature Chemical Biology

Year:

2015

Language:

english

File:

PDF, 97 KB

english, 2015

24

P1-419 In vivo characterization of LY450139, a novel, stereoselective, functional gamma-secretase inhibitor

Leonard N. Boggs, Kimberly S. Fuson, Bruce D. Gitter, Daniel L. Czilli, Paul A. Hyslop, Mark H. Bender, Weiying Li, James E. Audia, Jeffrey S. Nissen, Thomas E. Mabry, Binhui Ni, Yuan Su, Patrick C. M

Journal:

Neurobiology of Aging

Year:

2004

Language:

english

File:

PDF, 168 KB

english, 2004

25

Diels-alder cyclization of 2,8,10-undecatrienals as a route to 1,2,3,4,4a,5,6,8a-octahydronaphthalenes

James A. Marshall, James E. Audia, Jonathan Grote, Barry G. Shearer

Journal:

Year:

1986

Language:

english

File:

PDF, 1.04 MB

english, 1986

26

Synthesis and 5α-reductase inhibitory activity of 8-substituted benzo[ƒ]quinolinones derived from palladium mediated coupling reactions

Edward C.R. Smith, Loretta A. McQuaid, Robin L. Goode, Ann M. McNulty, Blake Lee Neubauer, Vincent P. Rocco, James E. Audia

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1998

Language:

english

File:

PDF, 205 KB

english, 1998

27

5-HT1F receptor agonists inhibit neurogenic dural inflammation in guinea pigs

Johnson, Kirk W., Schaus, John M., Durkin, Margaret M., Audia, James E., Kaldor, Stephen W., Flaugh, Michael E., Adham, Nika, Zgombick, John M., Cohen, Marlene L., Branchek, Theresa A., Phebus, Lee A.

Journal:

Year:

1997

Language:

english

File:

PDF, 400 KB

english, 1997

28

Encyclopedia of Reagents for Organic Synthesis || Dimethyl Diazomalonate

Audia, James E.

Year:

2001

Language:

english

File:

PDF, 152 KB

english, 2001

29

The Highly Selective Caspase-1 Inhibitor VX-765 Provides Additive Protection Against Myocardial Infarction in Rat Hearts When Combined With a Platelet Inhibitor

Yang, Xi-Ming, Downey, James M., Cohen, Michael V., Housley, Nicole A., Alvarez, Diego F., Audia, Jonathon P.

Journal:

Journal of Cardiovascular Pharmacology and Therapeutics

Year:

2017

Language:

english

File:

PDF, 182 KB

english, 2017

30

Acyclic stereocontrol in catalyzed intramolecular Diels-Alder cyclizations leading to octahydronaphthalenecarboxaldehydes

Marshall, James A., Grote, Jonathan, Audia, James E.

Journal:

Journal of the American Chemical Society

Year:

1987

Language:

english

File:

PDF, 1.22 MB

english, 1987

31

Encyclopedia of Reagents for Organic Synthesis || Dimethyl Diazomalonate

Audia, James E.

Year:

2001

Language:

english

File:

PDF, 115 KB

english, 2001

32

Responses of LNCaP prostatic adenocarcinoma cell cultures to LY300502, a benzoquinolinone human type I 5α-reductase inhibitor

Sutkowski, Debra M., Audia, James E., Goode, Robin L., Hsiao, Kenneth C., Leibovitch, Ilan Y., McNulty, Ann M., Neubauer, Blake Lee

Journal:

Year:

1996

Language:

english

File:

PDF, 428 KB

english, 1996

33

Improved Preparation of (E)-3-Trimethylsilyl-2-Buten-1-OL

Audia, James E., Marshall, James A.

Journal:

Synthetic Communications

Year:

1983

Language:

english

File:

PDF, 172 KB

english, 1983

34

Nonsteroidal inhibitors of human type I steroid 5-.alpha.-reductase

Jones, Charles D., Audia, James E., Lawhorn, David E., McQuaid, Loretta A., Neubauer, Blake L., Pike, Andrew J., Pennington, Pamela A., Stamm, Nancy B., Toomey, Richard E., Hirsch, Kenneth S.

Journal:

Journal of Medicinal Chemistry

Year:

1993

Language:

english

File:

PDF, 292 KB

english, 1993

35

Synthesis of two useful, enantiomerically pure derivatives of (S)-4-hydroxy-2-cyclohexenone

Audia, James E., Boisvert, Louise, Patten, Arthur D., Villalobos, Anabella, Danishefsky, Samuel J.

Journal:

Journal of Organic Chemistry

Year:

1989

Language:

english

File:

PDF, 436 KB

english, 1989

36

Building a Methodological Foundation for Impactful Urban Planetary Health Science

Pineo, Helen, Audia, Camilla, Black, Daniel, French, Matthew, Gemmell, Emily, Lovasi, Gina S., Milner, James, Montes, Felipe, Niu, Yanlin, PÃ©rez-Ferrer, Carolina, Siri, JosÃ©, Taruc, Ruzka R.

Journal:

Journal of Urban Health

Year:

2020

File:

PDF, 331 KB

2020

37

Irritable bowel syndrome: Present and prospective pharmacological intervention

William J. Kinnier, James F. Kachur, Vicki H. Audia, Carl Kaiser

Journal:

Medicinal Research Reviews

Year:

1989

Language:

english

File:

PDF, 1.02 MB

english, 1989

38

QSAR study of benzoquinolinones as inhibitors of human type 1 5-α-reductase.

James H. Wikel, Kerry G. Bemis, James E. Audia, Loretta A. McQuaid, Charles D. Jones, Pamela A. Pennington, David E. Lawhorn, Kenneth R. Hirsch, Nancy B. Stamm

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1993

Language:

english

File:

PDF, 425 KB

english, 1993

39

Encyclopedia of Reagents for Organic Synthesis || α-Diazoacetophenone

Audia, James E.

Year:

2001

Language:

english

File:

PDF, 63 KB

english, 2001

40

LY191704: A Selective, Nonsteroidal Inhibitor of Human Steroid 5α- Reductase Type 1

Kenneth S. Hirsch, Charles D. Jones, James E. Audia, Stefan Andersson, Loretta McQuaid, Nancy B. Stamm, Blake L. Neubauer, Pam Pennington, Richard E. Toomey and David W. Russell

Journal:

Proceedings of the National Academy of Sciences

Year:

1993

Language:

english

File:

PDF, 988 KB

english, 1993

41

Mentoring Matters in Drug Discovery

Blanco, Maria-Jesus, Audia, James E.

Journal:

ACS Medicinal Chemistry Letters

Year:

2020

File:

PDF, 623 KB

2020

42

A diastereoselective tandem metalloenamine alkylation/aza-annulation of β-tetralones expedites the synthesis of benzoquinolinones

James E. Audia, James J. Droste, James M. Dunigan, John Bowers, Perry C. Heath, Dale W. Holme, Jill H. Eifert, Harry A. Kay, Richard D. Miller, Jorge M. Olivares, Thomas F. Rainey, Leland O. Weigel

Journal:

Tetrahedron Letters

Year:

1996

Language:

english

File:

PDF, 220 KB

english, 1996

43

Potent, Selective Tetrahydro-β-carboline Antagonists of the Serotonin 2B (5HT2B) Contractile Receptor in the Rat Stomach Fundus

Audia, James E., Evrard, Deborah A., Murdoch, Gwyn R., Droste, James J., Nissen, Jeffrey S., Schenck, Kathy W., Fludzinski, Pawel, Lucaites, Virginia L., Nelson, David L., Cohen, Marlene L.

Journal:

Journal of Medicinal Chemistry

Year:

1996

Language:

english

File:

PDF, 297 KB

english, 1996

44

Discovery, Design, and Optimization of Isoxazole Azepine BET Inhibitors

Gehling, Victor S., Hewitt, Michael C., Vaswani, Rishi G., Leblanc, Yves, Côté, Alexandre, Nasveschuk, Christopher G., Taylor, Alexander M., Harmange, Jean-Christophe, Audia, James E., Pardo, Eneida,

Journal:

ACS Medicinal Chemistry Letters

Year:

2013

Language:

english

File:

PDF, 397 KB

english, 2013

45

GNE-886: A Potent and Selective Inhibitor of the Cat Eye Syndrome Chromosome Region Candidate 2 Bromodomain (CECR2)

Crawford, Terry D., Audia, James E., Bellon, Steve, Burdick, Daniel J., Bommi-Reddy, Archana, Côté, Alexandre, Cummings, Richard T., Duplessis, Martin, Flynn, Elizabeth Megan, Hewitt, Michael C., Huan

Journal:

ACS Medicinal Chemistry Letters

Year:

2017

Language:

english

File:

PDF, 920 KB

english, 2017

46

“Pictet-Spengler-like” Synthesis of Tetrahydro-β-carbolines under Hydrolytic Conditions. Direct Use of Azalactones as Phenylacetaldehyde Equivalents

Audia, James E., Droste, James J., Nissen, Jeffrey S., Murdoch, Gwyn L., Evrard, Deborah A.

Journal:

Journal of Organic Chemistry

Year:

1996

Language:

english

File:

PDF, 118 KB

english, 1996

47

Discovery of Benzotriazolo[4,3- d ][1,4]diazepines as Orally Active Inhibitors of BET Bromodomains

Taylor, Alexander M., Vaswani, Rishi G., Gehling, Victor S., Hewitt, Michael C., Leblanc, Yves, Audia, James E., Bellon, Steve, Cummings, Richard T., Côté, Alexandre, Harmange, Jean-Christophe, Jayara

Journal:

ACS Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 667 KB

english, 2015

48

The promise and peril of chemical probes

Arrowsmith, Cheryl H, Audia, James E, Austin, Christopher, Baell, Jonathan, Bennett, Jonathan, Blagg, Julian, Bountra, Chas, Brennan, Paul E, Brown, Peter J, Bunnage, Mark E, Buser-Doepner, Carolyn, C

Journal:

Nature Chemical Biology

Year:

2015

Language:

english

File:

PDF, 736 KB

english, 2015

49

Addition of n-butylcuprates to .alpha.-methylenecycloalkylidene epoxides

Marshall, James A., Audia, Vicki H.

Journal:

Journal of Organic Chemistry

Year:

1985

Language:

english

File:

PDF, 765 KB

english, 1985

50

Preparation and biological evaluation of conformationally constrained BACE1 inhibitors

Winneroski, Leonard L., Schiffler, Matthew A., Erickson, Jon A., May, Patrick C., Monk, Scott A., Timm, David E., Audia, James E., Beck, James P., Boggs, Leonard N., Borders, Anthony R., Boyer, Robert

Journal:

Bioorganic & Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.25 MB

english, 2015

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